CNS 11: Introduction to Benzodiazepines
Benzodiazepines (BZDs) Fact Sheet: Mechanism of Action: Potentiate activity of GABA at GABAa receptors. This leads to anxiolytic and sedating effects. *Pause* Does this make sense? GABA is an inhibitory neurotransmitter. BZDs increase the activity of GABA, which means more inhibitory effects. This leads to a sedating effect. Onset ofContinue Reading